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Nitric oxide induces the distinct invisibility phenotype of Mycobacterium tuberculosis.
Gap-Gaupool B, Glenn SM, Milburn E, Turapov O, Crosatti M, Hincks J, Stewart B, Bacon J, Kendall SL, Voskuil MI, Riabova O, Monakhova N, Green J, Waddell SJ, Makarov VA, Mukamolova GV
Commun Biol, 7(1):1206, 28 Sep 2024
Cited by: 0 articles | PMID: 39342050 | PMCID: PMC11439070
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Dynamic features of virus protein 1 and substitutions in the 3-phenyl ring determine the potency and broad-spectrum activity of capsid-binding pyrazolo[3,4-d]pyrimidines against rhinoviruses.
Richter M, Khrenova M, Kazakova E, Riabova O, Egorova A, Makarov V, Schmidtke M
Antiviral Res, 231:105993, 03 Sep 2024
Cited by: 0 articles | PMID: 39233314
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The novel drug candidate VOMG kills Mycobacterium abscessus and other pathogens by inhibiting cell division.
Degiacomi G, Chiarelli LR, Riabova O, Loré NI, Muñoz-Muñoz L, Recchia D, Stelitano G, Postiglione U, Saliu F, Griego A, Scoffone VC, Kazakova E, Scarpa E, Ezquerra-Aznárez JM, Stamilla A, Buroni S, Tortoli E, Rizzello L, Sassera D, [...] Pasca MR
Int J Antimicrob Agents, 64(4):107278, 26 Jul 2024
Cited by: 0 articles | PMID: 39069229
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Needle tracking in low-resolution ultrasound volumes using deep learning.
Grube S, Latus S, Behrendt F, Riabova O, Neidhardt M, Schlaefer A
Int J Comput Assist Radiol Surg, 19(10):1975-1981, 13 Jul 2024
Cited by: 0 articles | PMID: 39002100 | PMCID: PMC11442564
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Efficacy of macozinone in mice with genetically diverse susceptibility to Mycobacterium tuberculosis infection.
Nikonenko B, Logunova N, Egorova A, Kapina M, Sterzhanova N, Bocharova I, Kondratieva E, Riabova O, Semyonova L, Makarov V, Dedicated to the 10th anniversary of the iM4TB Foundation
Microbes Infect, 105376, 07 Jun 2024
Cited by: 0 articles | PMID: 38852904
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Characterization of the dispirotripiperazine derivative PDSTP as antibiotic adjuvant and antivirulence compound against Pseudomonas aeruginosa.
Bonacorsi A, Trespidi G, Scoffone VC, Irudal S, Barbieri G, Riabova O, Monakhova N, Makarov V, Buroni S
Front Microbiol, 15:1357708, 16 Feb 2024
Cited by: 0 articles | PMID: 38435690 | PMCID: PMC10904629
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SCRAPPY - a single cell rapid assay of proteome perturbation in yeast uncovers a joint role of aromatic amino acids and oxidative stress in the toxicity of lipophilic nucleoside analogs
Ghazy E, Bidiuk VA, Ryabov F, Mitkevich OV, Riabova OB, Stanishevskiy YM, Levshin IB, Alexandrova LA, Jasko MV, Makarov DA, Zhgun AA, Avdanina DA, Ermolyuk AA, Kushnirov VV, Egorova AP, Agaphonov MO, Alexandrov AI
bioRxiv, 20 Feb 2024
Cited by: 0 articles | PPR: PPR810700
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Molecular mechanism of rhinovirus escape from the Pyrazolo[3,4-d]pyrimidine capsid-binding inhibitor OBR-5-340 via mutations distant from the binding pocket: Derivatives that brake resistance.
Richter M, Döring K, Blaas D, Riabova O, Khrenova M, Kazakova E, Egorova A, Makarov V, Schmidtke M
Antiviral Res, 222:105810, 18 Jan 2024
Cited by: 0 articles | PMID: 38244889
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Antidepressant-like Effect of the Eburnamine-Type Molecule Vindeburnol in Rat and Mouse Models of Ultrasound-Induced Depression.
Zubkov E, Riabova O, Zorkina Y, Egorova A, Ushakova V, Lepioshkin A, Novoselova E, Abramova O, Morozova A, Chekhonin V, Makarov V
ACS Chem Neurosci, 15(3):560-571, 12 Jan 2024
Cited by: 0 articles | PMID: 38216514
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Determination of alkaloid-inspired molecule vindeburnol in rabbit plasma by UPLC-HRMS and its application to pharmacokinetic studies and preliminary metabolite identification.
Tsedilin A, Borets L, Riabova O, Kazakova E, Tafeenko V, Makarov V
J Pharm Biomed Anal, 239:115917, 13 Dec 2023
Cited by: 0 articles | PMID: 38101239
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1-Sulfonyl-3-amino-1H-1,2,4-triazoles as Yellow Fever Virus Inhibitors: Synthesis and Structure-Activity Relationship.
Kazakova E, Lane TR, Jones T, Puhl AC, Riabova O, Makarov V, Ekins S
ACS Omega, 8(45):42951-42965, 01 Nov 2023
Cited by: 0 articles | PMID: 38024733 | PMCID: PMC10653066
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Benzothiozinone derivatives with anti-tubercular Activity-Further side chain investigation.
Wu X, Wang W, Stelitano G, Riabova O, Wang B, Niu W, Cocorullo M, Shi R, Chiarelli LR, Makarov V, Lu Y, Li C, Qiao C
Eur J Med Chem, 264:115976, 25 Nov 2023
Cited by: 0 articles | PMID: 38039794
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Antiviral Evaluation of Dispirotripiperazines against Hepatitis B Virus.
Jones T, Tavis JE, Li Q, Riabova O, Monakhova N, Bradley DP, Lane TR, Makarov V, Ekins S
J Med Chem, 66(17):12459-12467, 23 Aug 2023
Cited by: 0 articles | PMID: 37611244 | PMCID: PMC11017374
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Efficacy of an isoxazole-3-carboxamide analog of pleconaril in mouse models of Enterovirus-D68 and Coxsackie B5.
Lane TR, Fu J, Sherry B, Tarbet B, Hurst BL, Riabova O, Kazakova E, Egorova A, Clarke P, Leser JS, Frost J, Rudy M, Tyler KL, Klose T, Volobueva AS, Belyaevskaya SV, Zarubaev VV, Kuhn RJ, Makarov V, Ekins S
Antiviral Res, 216:105654, 14 Jun 2023
Cited by: 2 articles | PMID: 37327878 | PMCID: PMC10527014
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Side Chain-Modified Benzothiazinone Derivatives with Anti-Mycobacterial Activity.
Fan D, Wang B, Stelitano G, Savková K, Riabova O, Shi R, Wu X, Chiarelli LR, Mikušová K, Makarov V, Lu Y, Hong Y, Qiao C
Biomedicines, 11(7):1975, 12 Jul 2023
Cited by: 0 articles | PMID: 37509615 | PMCID: PMC10377601
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N-Phenyl-1-(phenylsulfonyl)-1H-1,2,4-triazol-3-amine as a New Class of HIV-1 Non-nucleoside Reverse Transcriptase Inhibitor.
Lane T, Makarov V, Nelson JAE, Meeker RB, Sanna G, Riabova O, Kazakova E, Monakhova N, Tsedilin A, Urbina F, Jones T, Suchy A, Ekins S
J Med Chem, 66(9):6193-6217, 02 May 2023
Cited by: 4 articles | PMID: 37130343 | PMCID: PMC10269403
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Side Chain-modified Benzothiazinone Derivatives with Anti-Mycobacterial Activity
Dongguang F, Wang B, Stelitano G, Savková K, Riabova O, Shi R, Wu X, Chiarelli LR, Mikušová K, Makarov V, Lu Y, Hong Y, Qiao C
Preprints.org, 01 Jun 2023
Cited by: 0 articles | PPR: PPR669536
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Antituberculosis Macozinone Extended-Release Tablets To Enhance Bioavailability: a Pilot Pharmacokinetic Study in Beagle Dogs.
Koryakova A, Shcherbakova V, Riabova O, Kazaishvili Y, Bolgarin R, Makarov V
Microbiol Spectr, 11(1):e0232722, 12 Dec 2022
Cited by: 2 articles | PMID: 36507624 | PMCID: PMC9927148
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Multiple approaches to repurposing drugs for neuroblastoma.
Rank L, Puhl AC, Havener TM, Anderson E, Foil DH, Zorn KM, Monakhova N, Riabova O, Hickey AJ, Makarov V, Ekins S
Bioorg Med Chem, 73:117043, 04 Oct 2022
Cited by: 3 articles | PMID: 36208544 | PMCID: PMC9870653
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Thieno[2,3-d]pyrimidine-Core Compounds Show Activity against Clinically Relevant Gram-Positive Bacteria.
Riabova O, Egorova A, Lepioshkin A, Li Y, Voigt K, Kloss F, Makarov V
ChemMedChem, 17(17):e202200207, 09 Aug 2022
Cited by: 0 articles | PMID: 35880634
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A proof-of-concept study for the efficacy of dispirotripiperazine PDSTP in a rabbit model of herpes simplex epithelial keratitis.
Alimbarova L, Egorova A, Riabova O, Monakhova N, Makarov V
Antiviral Res, 202:105327, 27 Apr 2022
Cited by: 4 articles | PMID: 35487465
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Pyronaridine Protects against SARS-CoV-2 Infection in Mouse.
Puhl AC, Gomes GF, Damasceno S, Godoy AS, Noske GD, Nakamura AM, Gawriljuk VO, Fernandes RS, Monakhova N, Riabova O, Lane TR, Makarov V, Veras FP, Batah SS, Fabro AT, Oliva G, Cunha FQ, Alves-Filho JC, Cunha TM, Ekins S
ACS Infect Dis, 8(6):1147-1160, 24 May 2022
Cited by: 18 articles | PMID: 35609344
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Machine Learning Models for Mycobacterium tuberculosisIn Vitro Activity: Prediction and Target Visualization.
Lane TR, Urbina F, Rank L, Gerlach J, Riabova O, Lepioshkin A, Kazakova E, Vocat A, Tkachenko V, Cole S, Makarov V, Ekins S
Mol Pharm, 19(2):674-689, 29 Dec 2021
Cited by: 9 articles | PMID: 34964633 | PMCID: PMC9121329
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Strain dependent structural effects and in vivo efficacy of enterovirus-D68 inhibitors
Lane T, Fu J, Sherry B, Tarbet B, Hurst BL, Riabova O, Kazakova E, Egorova A, Clarke P, Leser JS, Frost J, Rudy M, Tyler K, Klose T, Kuhn RJ, Makarov V, Ekins S
bioRxiv, 27 Dec 2021
Cited by: 0 articles | PPR: PPR436994
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Pyronaridine Protects Against SARS-CoV-2 in Mouse
Puhl AC, Gomes GF, Damasceno S, Godoy AS, Noske GD, Nakamura AM, Gawriljuk VO, Fernandes RS, Monakhova N, Riabova O, Lane TR, Makarov V, Veras FP, Batah SS, Fabro AT, Oliva G, Cunha FQ, Alves-Filho JC, Cunha TM, Ekins S
bioRxiv, 30 Sep 2021
Cited by: 0 articles | PPR: PPR402754
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1-25 of 67 results

1 2 3

Search life-sciences literature (45,103,589 articles, preprints and more)

Search results

Nitric oxide induces the distinct invisibility phenotype of Mycobacterium tuberculosis.

Dynamic features of virus protein 1 and substitutions in the 3-phenyl ring determine the potency and broad-spectrum activity of capsid-binding pyrazolo[3,4-d]pyrimidines against rhinoviruses.

The novel drug candidate VOMG kills Mycobacterium abscessus and other pathogens by inhibiting cell division.

Needle tracking in low-resolution ultrasound volumes using deep learning.

Efficacy of macozinone in mice with genetically diverse susceptibility to Mycobacterium tuberculosis infection.

Characterization of the dispirotripiperazine derivative PDSTP as antibiotic adjuvant and antivirulence compound against Pseudomonas aeruginosa.

SCRAPPY - a single cell rapid assay of proteome perturbation in yeast uncovers a joint role of aromatic amino acids and oxidative stress in the toxicity of lipophilic nucleoside analogs

Molecular mechanism of rhinovirus escape from the Pyrazolo[3,4-d]pyrimidine capsid-binding inhibitor OBR-5-340 via mutations distant from the binding pocket: Derivatives that brake resistance.

Antidepressant-like Effect of the Eburnamine-Type Molecule Vindeburnol in Rat and Mouse Models of Ultrasound-Induced Depression.

Determination of alkaloid-inspired molecule vindeburnol in rabbit plasma by UPLC-HRMS and its application to pharmacokinetic studies and preliminary metabolite identification.

1-Sulfonyl-3-amino-1H-1,2,4-triazoles as Yellow Fever Virus Inhibitors: Synthesis and Structure-Activity Relationship.

Benzothiozinone derivatives with anti-tubercular Activity-Further side chain investigation.

Antiviral Evaluation of Dispirotripiperazines against Hepatitis B Virus.

Efficacy of an isoxazole-3-carboxamide analog of pleconaril in mouse models of Enterovirus-D68 and Coxsackie B5.

Side Chain-Modified Benzothiazinone Derivatives with Anti-Mycobacterial Activity.

N-Phenyl-1-(phenylsulfonyl)-1H-1,2,4-triazol-3-amine as a New Class of HIV-1 Non-nucleoside Reverse Transcriptase Inhibitor.

Side Chain-modified Benzothiazinone Derivatives with Anti-Mycobacterial Activity

Antituberculosis Macozinone Extended-Release Tablets To Enhance Bioavailability: a Pilot Pharmacokinetic Study in Beagle Dogs.

Multiple approaches to repurposing drugs for neuroblastoma.

Thieno[2,3-d]pyrimidine-Core Compounds Show Activity against Clinically Relevant Gram-Positive Bacteria.

A proof-of-concept study for the efficacy of dispirotripiperazine PDSTP in a rabbit model of herpes simplex epithelial keratitis.

Pyronaridine Protects against SARS-CoV-2 Infection in Mouse.

Machine Learning Models for Mycobacterium tuberculosisIn Vitro Activity: Prediction and Target Visualization.

Strain dependent structural effects and in vivo efficacy of enterovirus-D68 inhibitors

Pyronaridine Protects Against SARS-CoV-2 in Mouse

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