Altered fibroblast growth factor receptor 4 stability promotes prostate cancer progression

Neoplasia. 2008 Aug;10(8):847-56. doi: 10.1593/neo.08450.

Abstract

Fibroblast growth factor receptor 4 (FGFR-4) is expressed at significant levels in almost all human prostate cancers, and expression of its ligands is ubiquitous. A common polymorphism of FGFR-4 in which arginine (Arg(388)) replaces glycine (Gly(388)) at amino acid 388 is associated with progression in human prostate cancer. We show that the FGFR-4 Arg(388) polymorphism, which is present in most prostate cancer patients, results in increased receptor stability and sustained receptor activation. In patients bearing the FGFR-4 Gly(388) variant, expression of Huntingtin-interacting protein 1 (HIP1), which occurs in more than half of human prostate cancers, also results in FGFR-4 stabilization. This is associated with enhanced proliferation and anchorage-independent growth in vitro. Our findings indicate that increased receptor stability and sustained FGFR-4 signaling occur in most human prostate cancers due to either the presence of a common genetic polymorphism or the expression of a protein that stabilizes FGFR-4. Both of these alterations are associated with clinical progression in patients with prostate cancer. Thus, FGFR-4 signaling and receptor turnover are important potential therapeutic targets in prostate cancer.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, Non-P.H.S.

MeSH terms

  • DNA-Binding Proteins / genetics*
  • DNA-Binding Proteins / metabolism
  • Disease Progression
  • Fibroblast Growth Factor 2 / genetics
  • Gene Expression Regulation, Neoplastic / genetics*
  • Genetic Variation / drug effects
  • Genetic Variation / genetics
  • Humans
  • Ligands
  • Male
  • Phosphorylation
  • Polymorphism, Genetic / genetics
  • Prostatic Neoplasms / genetics*
  • Prostatic Neoplasms / metabolism
  • Prostatic Neoplasms / pathology*
  • RNA, Messenger / genetics
  • Receptor, Fibroblast Growth Factor, Type 4 / drug effects
  • Receptor, Fibroblast Growth Factor, Type 4 / genetics*
  • Receptor, Fibroblast Growth Factor, Type 4 / metabolism

Substances

  • DNA-Binding Proteins
  • HIP1 protein, human
  • Ligands
  • RNA, Messenger
  • Fibroblast Growth Factor 2
  • FGFR4 protein, human
  • Receptor, Fibroblast Growth Factor, Type 4