The effect of PPARγ inhibition on bone marrow adipose tissue and bone in C3H/HeJ mice

Am J Physiol Endocrinol Metab. 2019 Jan 1;316(1):E96-E105. doi: 10.1152/ajpendo.00265.2018. Epub 2018 Nov 20.

Abstract

Bone marrow adipose tissue (BMAT) increases after menopause, and increased BMAT is associated with osteoporosis and prevalent vertebral fractures. Peroxisome proliferator-activated receptor-γ (PPARγ) activation promotes adipogenesis and inhibits osteoblastogenesis; therefore, PPARγ is a potential contributor to the postmenopausal increase in BMAT and decrease in bone mass. The aim of this study is to determine if PPARγ inhibition can prevent ovariectomy-induced BMAT increase and bone loss in C3H/HeJ mice. Fourteen-week-old female C3H/HeJ mice ( n = 40) were allocated to four intervention groups: sham surgery (Sham) or ovariectomy (OVX; isoflurane anesthesia) with either vehicle (Veh) or PPARγ antagonist administration (GW9662; 1 mg·kg-1·day-1, daily intraperitoneal injections) for 3 wk. We measured BMAT volume, adipocyte size, adipocyte number. and bone structural parameters in the proximal metaphysis of the tibia using polyoxometalate-based contrast enhanced-nanocomputed topogaphy. Bone turnover was measured in the contralateral tibia using histomorphometry. The effects of surgery and treatment were analyzed by two-way ANOVA. OVX increased the BMAT volume fraction (Sham + Veh: 2.9 ± 2.7% vs. OVX + Veh: 8.1 ± 5.0%: P < 0.001), average adipocyte diameter (Sham + Veh: 19.3 ± 2.6 μm vs. OVX + Veh: 23.1 ± 3.4 μm: P = 0.001), and adipocyte number (Sham + Veh: 584 ± 337cells/μm3 vs. OVX + Veh: 824 ± 113cells/μm3: P = 0.03), while OVX decreased bone volume fraction (Sham + Veh: 15.5 ± 2.8% vs. OVX + Veh: 7.7 ± 1.9%; P < 0.001). GW9662 had no effect on BMAT, bone structural parameters, or bone turnover. In conclusion, ovariectomy increased BMAT and decreased bone volume in C3H/HeJ mice. The PPARγ antagonist GW9662 had no effect on BMAT or bone volume in C3H/HeJ mice, suggesting that BMAT accumulation is regulated independently of PPARγ in C3H/HeJ mice.

Keywords: C3H/HeJ mice; PPARγ antagonist; bone marrow adipose tissue; bone turnover; ovariectomy.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adipocytes / drug effects*
  • Adipocytes / pathology
  • Adipose Tissue / drug effects*
  • Adipose Tissue / pathology
  • Anilides / pharmacology*
  • Animals
  • Bone Marrow / drug effects*
  • Bone Marrow / pathology
  • Bone Remodeling / drug effects
  • Cell Count
  • Cell Size
  • Female
  • Humans
  • Mice
  • Mice, Inbred C3H
  • Organ Size
  • Osteoporosis, Postmenopausal
  • Ovariectomy
  • PPAR gamma / antagonists & inhibitors*
  • Tibia / diagnostic imaging
  • Tibia / drug effects*
  • Tomography, X-Ray Computed

Substances

  • 2-chloro-5-nitrobenzanilide
  • Anilides
  • PPAR gamma