http://rdf.ncbi.nlm.nih.gov/pubchem/patent/EP-1565450-B1
Outgoing Links
| Predicate | Object |
|---|---|
| assignee | http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_eccd894c99fea2d1c0c8735872bb2309 |
| classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D309-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D309-06 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D309-08 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D309-30 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D409-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D309-20 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D407-06 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D409-08 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D407-12 |
| classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D309-30 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D309-06 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D309-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D309-08 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D409-08 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D309-20 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D409-04 |
| filingDate | 2003-11-17^^<http://www.w3.org/2001/XMLSchema#date> |
| grantDate | 2007-07-04^^<http://www.w3.org/2001/XMLSchema#date> |
| inventor | http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_eb221f66072f414bccd3b7d87c165692 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_6d9c82eb04894bf2555523406eb0aa1c http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_fbcf75a75b2155fc46cbaa5223543cdf http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_4a8d8c514adf7dd10c5c8abf6bf717f7 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_afa18e11d1f39609eba94717b7062bb0 |
| publicationDate | 2007-07-04^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber | EP-1565450-B1 |
| titleOfInvention | Tetrahydropyran derivatives |
| abstract | 2,5-Di-substituted tetrahydropyran derivatives (I) are new. 2,5-Di-substituted tetrahydropyran derivatives of formula (I) are new: R11 = H, F, Cl, Br, I, CN, aryl, heterocyclyl or Alk; Alk = optionally halogenated 1-15C alkyl (where CH2 group(s) is optionally replaced by -C triple bond C-, -CH=CH-, O, CO, COO or OCO); A = Cyc, tetrahydropyran-2,5-diyl, 1,3-dioxan-2,5-diyl or pyrimidine-2,5-diyl; Cyc = trans-1,4-cyclohexylene; a = 0 - 2; Z11 = bond, -CH2CH2-, -CF2CF2-, -CF2CH2-, -CH2CF2-, -CH2O-, -OCH2-, -CF2O- or -OCF2-; W = CH- or C=; B, D = Cyc, 4-cyclohexylidene-1-yl (Cyc=) or ArL; ArL = 1,4-phenylene (substituted with L1, L2 and L3 at positions 3, 5 and 6); b, d = 0 or 1; Y11 = =O, =C(SR12)(SR13), =CF2, H, F, Cl, Br, I, CN, OH, SH, -COR14, -OSO2R15, -C(=S+R12)(-SR13)X-, -B(OR16)(OR17), -BF3- Cat+, -Si(OR18)(OR19)(OR20) or Alk; Y12, Y13 = H or Alk; L1 - L3 = H or F; R12, R13 = 1-15C alkyl; or R12+R13 = -(CH2)p- in which 1, 2 or 3 of the CH2 groups may be substituted with 1-8C alkyl group(s); p = 2 - 6; R14 = OH, aryl(oxy), alkoxy, aralkoxy, Cl, Br, aralkyl or alkyl; R15 = aryl, aralkyl or Alk; R16, R17 = H or 1-15C alkyl; or R16+R17 = -(CH2)p- in which 1, 2 or 3 of the CH2 groups may be substituted with 1-8C alkyl group(s); R18 - R20 = 1-15C alkyl; Cat = alkali metal or quaternary ammonium cation; X = weakly-coordinating anion; and provided that: (i) if W is -ArL-(ArL)d-Y11, then Y11 is H, I, OH, SH, -COOR14, -OSO2R15, -C(=S+R12)(SR13)X-, -B(OR16)(OR17), -BF3- Cat+, -Si(OR18)(OR19)(OR20) or Alk (excluding alkoxy); (ii) if b+d is not zero, then W is CH-; (iii) if B or D is ArL, then Y11 is not O, =C(SR12)(SR13) or =CF2; (iv) if d is 1, then B is not Cyc; and (v) if a is 2, then A can have different meanings (undefined). Independent claims are also included for methods (M1) - (M5) for the production of compounds of formula (IA), (IB), (IC), (ID) and (IE), respectively. R11' = H, F, Cl, Br, I, CN, aryl, heterocyclyl or alkyl; Y12', Y13' = H or alkyl; Y11' = =O, =C(SR12)(SR13) or =CF2; Y11'' = H, F, Cl, Br, I, CN, OH or -B(OR16)(OR17); and Y11''' = -COOH or -C(=S+R12)(SR13)X-. |
| priorityDate | 2002-11-27^^<http://www.w3.org/2001/XMLSchema#date> |
| type | http://data.epo.org/linked-data/def/patent/Publication |
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