http://rdf.ncbi.nlm.nih.gov/pubchem/patent/EP-3310765-A1
Outgoing Links
| Predicate | Object |
|---|---|
| assignee | http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_c83971dae1af3500e88babcc816556a3 |
| classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D243-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/B01J31-24 |
| classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D243-10 |
| filingDate | 2016-06-21^^<http://www.w3.org/2001/XMLSchema#date> |
| inventor | http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_68abaf09a882744b446262ee626b8670 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_51d231248ac672eeebabfebf5ae2c37c |
| publicationDate | 2018-04-25^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber | EP-3310765-A1 |
| titleOfInvention | Process for preparing 1,4-dibenzodiazepines via buchwald-hartwig chemistry |
| abstract | The present application provides a one-pot catalytic process which involves the formation of 1,4-dibenzodiazepines from o-haloaldimines (either pre-formed or formed in situ ) of formula (I) and o-haloanilines of formula (II) via a palladium catalyzed Buchwald-Hartwig reaction and a cyclization sequence, to afford the 1,4-dibenzodiazepine products of formula (III). The present application describes the preparation of the 1,4-dibenzodiazepine products of formula (III) from simple commercial raw materials by efficient processes. |
| priorityDate | 2015-06-22^^<http://www.w3.org/2001/XMLSchema#date> |
| type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
Showing number of triples: 1 to 167 of 167.