http://rdf.ncbi.nlm.nih.gov/pubchem/patent/ES-2357015-T3
Outgoing Links
| Predicate | Object |
|---|---|
| assignee | http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_d5cd84f92e5e2ff95dfd19e4e329db3b |
| classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D277-82 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P3-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P3-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P3-06 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P3-08 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P3-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D263-58 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D235-30 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P43-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D513-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P5-50 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P9-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P9-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P7-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P9-00 |
| classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P3-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D513-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D277-82 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-428 |
| filingDate | 2005-10-14^^<http://www.w3.org/2001/XMLSchema#date> |
| grantDate | 2011-04-15^^<http://www.w3.org/2001/XMLSchema#date> |
| inventor | http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_d92b07d94b190f7cafbf62c84d246e5c http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_9cc783621b51ba298190ab753dff5ea3 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_be7771337f4cac2366a64aa4f47fe5c4 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_c3030f58eba62754c156604c5f0bd997 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_21ce2091474b34c98983b3db399942e9 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_4e153241469fb543a00f206b6e9483d9 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_df4d05298e56c9848e7b2efdc9092dc4 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_8443d270e9bf88f7e8df3a012048105d http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_68cfbfe15e68f3af38385f0ab6c11573 |
| publicationDate | 2011-04-15^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber | ES-2357015-T3 |
| titleOfInvention | PREPARATION AND USE OF BIFENIL-4-ILCARBONYLAMINO ACID DERIVATIVES FOR THE TREATMENT OF OBESITY. |
| abstract | A compound of formula (I) ** Formula ** in which Q is O, NR11, or S; it is a condensed ring selected from an aromatic 6-membered ring containing 0 or 1 N atoms; R1 is independently selected from halogen, (C1-C6) alkyl, (C1-C6) alkoxy, nitro, cyano, halo (C1-C6) alkyl, halo (C1-C6) haloalkoxy, aminocarbonyl, ((C1-C6) alkyl) aminocarbonyl , bis [(C1-C6) alkyl] aminocarbonyl, aminosulfonyl, ((C1-C6) alkyl) aminosulfonyl, bis [C1-C6 alkyl]] aminosulfonyl, ((C1-C6) alkyl) carbonylamino, (C1- alkyl C6)) sulfonyl, ((C1-C6) alkyl) sulfonylamino, hydroxy ((C1-C6) alkyl) aminocarbonyl, 1-morpholinylcarbonyl, and 1- piperidinylcarbonyl, and when two of said R1 substituents are (C1-C6) alkyl and they are attached to adjacent carbon atoms of ring A, they can be joined to form a 5-7 membered carbocyclic ring; n is 0, 1 or 2; R2 and R3 are independently selected from hydrogen, halogen, hydroxy, (C1-C6) alkyl, trifluoromethyl, (C1-C6) alkoxy, and trifluoromethoxy; R4 is selected from ** Formula ** in which R6 is H or CH3; and R7 is ** Formula ** in which R9 is selected from (C1-C6) alkyl optionally substituted with one or two groups selected from vinyl, CF3, OH, methoxy, SCH3, NH2, -CO2H, and -CONH2, ( CH2) mphenyl, in which m is 0 to 3, and in which the phenyl ring is optionally substituted with one or two groups selected from halogen, (C1-C6) alkyl, (C1-C6) alkoxy, OH, nitro, and cyano, piperidinyl optionally substituted in C with halogen, and optionally substituted in C or N with (C1-C6) alkyl, (C1-C6) alkoxy, nitro, or cyano, tetrahydropyran-4-yl; R10 is H or methyl; or R9 and R10 may form, together with the carbon to which they are attached, a 3- to 6-membered carbocyclic ring, R8 is hydrogen, (C1-C4) alkyl, hydroxy, or methoxy; R5 is selected from H, (C1-C6) alkyl, and hydroxy ((C2-C6) alkyl); R11 is selected from H, (C1-C6) alkyl, and hydroxy ((C2-C6) alkyl); and its pharmaceutically acceptable esters and salts. |
| priorityDate | 2004-10-15^^<http://www.w3.org/2001/XMLSchema#date> |
| type | http://data.epo.org/linked-data/def/patent/Publication |
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