abstract |
THE COMPOUNDS ARE 2,1-BENZISOTHIAZOLINE - 2,2-DIOXIDES SUBSITUTED IN THE 5-POSITION BY A 2-MOROPHOLINYL GROUP. THE COMPOUNDS ARE USEFUL AS CENTRAL NERVOUS SYSTEM DEPRESSANTS. THE COMPOUNDS MAY ALSO BE USED AS INTERMEDIATES IN THE PREPARATION OF PICKLING AGENTS, MOTHPROOFING AGENTS AND WOOD PRESERVATIVES. COMPOUNDS DISCLOSED INCLUDE 1-METHYL-5-(4-BENZYL-5/OXO - 2 - MORPHOLINYL)-2,1BENZIOTHIAZOLINE - 2,2 - DIOXIDE, 1-METHYL-5-(4-BENZYL-2MORPHOLINYL)-2,1-BENZISOTHIAZOLINE - 2,2 - DIOXIDE HYDROCHLORIDE, AND 1-METHYL-5-(2-MORPHALINYL) - 2,1 - BENZISOTHIAZOLINE-2,2-DIOXIDE HYDROCHLORIDE. |